THERAPEUTIC AREA PORTFOLIO · 44 PRODUCTS
Cardiovascular & Hematology
心血管与血液疾病
This portfolio supports anticoagulant and antiplatelet programs, lipid-lowering therapies, heart-failure and cardiomyopathy candidates, and selected hematology programs represented by the catalog’s terminal APIs.
Target APIs & Active Pipeline Programs in Cardiovascular & Hematology
EdoxabanMilvexianTicagrelorVoxelotorAtorvastatin calciumMK-0616ApixabanEzetimibeFostamatinibIptacopan HClObicetrapibRivaroxabanVericiguatBaxdrostatFinerenoneIndapamideLercanidipineNicardipineMavacamten
Cardiovascular & Hematology Products (44)
Catalog products related to terminal APIs in this area.
A-01CAS 545445-44-1
5,6-Dihydro-3-(4-morpholinyl)-1-[4-(2-oxo-1-piperidinyl)phenyl]-2(1H)-pyridinoneTarget API: Apixaban
A-03CAS 125971-94-0
(4R,6R)-tert-Butyl-6-cyanomethyl-2,2-dimethyl-1,3-dioxane-4-acetateTarget API: Atorvastatin calcium
A-04CAS 1146629-84-6
(R)-3-cyclopentyl-3-(4-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1H-pyrazol-1-yl)propanenitrileTarget API: Atorvastatin calcium
A-05CAS 125971-96-2
2-[2-(4-Fluorophenyl)-2-oxo-1-phenylethyl]-4-methyl-3-oxo-N-phenylpentanamideTarget API: Atorvastatin calcium
A-06CAS 147118-36-3
4-(4-Fluorophenyl)-6-Isopropyl-2-[ (N-Methyl-N-Methylsulfonyl) Amino]Pyrimidine-5-YL-MethanolTarget API: Atorvastatin calcium
A-07CAS 720720-96-7
5-Methyl-6,7-dihydro-4H-[1,3]thiazolo[5,4-c]pyridine-2- carboxylic acid;hydrochlorideTarget API: Edoxaban
A-08CAS 365997-33-7
Ethyl (1S,3R,4R)-4-hydroxy-3-[(2-methylpropan-2-yl) oxycarbonylamino]cyclohexane-1-carboxylateTarget API: Edoxaban
A-10CAS 1243308-37-3
Ethyl 2-[(5-chloropyridin-2-yl)amino]-2-oxoacetate; hydrochlorideTarget API: Edoxaban
A-11CAS 1210348-34-7
Tert-butyl N-[(1R,2S,5S)-2-Amino-5-(dimethylcarbamoyl) cyclohexyl]carbamate;oxalic acidTarget API: Edoxaban
A-12CAS 365998-36-3
Tert-butyl N-[(1R,2S,5S)-2-amino-5-(Dimethylcarbamoyl) cyclohexyl]carbamateTarget API: Edoxaban
A-13CAS 189028-95-3
(4S)-3-[(5S)-5-(4-fluorophenyl)-5-hydroxypentanoyl]-4-phenyl-1,3-oxazolidin-2-oneTarget API: Ezetimibe
A-18CAS 74936-72-4
5-(Methoxycarbonyl)-2,6-dimethyl-4-(3-nitrophenyl)-1,4-dihydropyridine-3-carboxylic acidTarget API: Lercanidipine/Nicardipine
A-19CAS 908846-88-8
(S)-2-((((9H-Fluoren-9-yl)methoxy)carbonyl)amino)-3-(5-fluoro-1H-indol-3-yl)propanoic acidTarget API: MK-0616
A-22CAS 94790-24-6
(S)-2-tertButoxycarbonylamino-3-(4-methoxy-phenyl)-propionic acid methyl esterTarget API: MK-0616
A-33CAS 376608-71-8
(1R,2S)-2-(3,4-Difluorophenyl)cyclopropanaminium (2R)-hydroxy(phenyl)ethanoateTarget API: Ticagrelor
A-34CAS 1156491-10-9
(1R,2S)-rel-2-(3,4-Difluorophenyl)cyclopropanamine hydrochlorideTarget API: Ticagrelor
A-35CAS 376608-65-0
2-[[(3aR,4S,6R,6aS)-6-Aminotetrahydro-2,2-dimethyl-4H-cyclopenta-1,3-dioxol-4-yl]oxy]-ethanol (2R,3R)-2,3-dihydroxybutanedioateTarget API: Ticagrelor
A-37CAS 1350653-26-7
5-fluoro-1-(2-fluorobenzyl)-1H-pyrazolo[3,4-b]pyridine-3-carbonitrileTarget API: Vericiguat
A-38CAS 1350653-24-5
5-fluoro-1-(2-fluorobenzyl)-3-iodo-1H-pyrazolo[3,4-b]pyridineTarget API: Vericiguat
A-39CAS 261947-64-2
Ethyl (2R,4S)-4-amino-2-ethyl-6-(trifluoromethyl)-3,4-dihydroquinoline-1(2H)-carboxylateTarget API: Obicetrapib
E-23CAS 1002726-62-6
6-Amino-2,2-Dimethyl-4H-Pyrido [3,2-B] [1,4] Oxazin-3-oneTarget API: Fostamatinib
E-45CAS 1481631-51-9
tert-Butyl 4-formyl-5-methoxy-7-methyl-1H-indole-1-carboxylateTarget API: Iptacopan HCl
H-16CAS 903550-26-5
(tetrahydro-2h-pyran-2-yl)-5-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)-1h-pyrazoleTarget API: Voxelotor
