THERAPEUTIC AREA PORTFOLIO · 52 PRODUCTS
Oncology
肿瘤
Our oncology portfolio follows the terminal APIs represented in the catalog, spanning kinase inhibitors, DNA-damage and cell-cycle programs, endocrine oncology, and building blocks for ADC and PROTAC development.
Target APIs & Active Pipeline Programs in Oncology
SelpercatinibCapmatinibBrigatinibElacestrantEntrectinibNiraparibTrilaciclibCamizestrantCapivasertibCarfilzomibEncorafenibPalbociclibAbemaciclibAdagrasibLorlatinibOsimertinibRibociclibSotorasibADC PayloadADC LinkerPROTAC Linker
Oncology Products (52)
Catalog products related to terminal APIs in this area.
C-06CAS 1197377-31-3
[2-Chloro-1-hydroxy-3-(6-quinolinyl)propyl]-2,5-pyrrolidinedioneTarget API: Capmatinib
C-12CAS 1013916-37-4
2-chloro-8-cyclopentyl-5-Methylpyrido[2,3-d]pyrimidin-7(8H)-oneTarget API: Palbociclib
C-13CAS 571188-59-5
tert-butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylateTarget API: Palbociclib
C-18CAS 1374635-90-1
Spiro[cyclohexane-1,9'(6'H)-pyrazino[1',2':1,5]pyrrolo[2,3-d] pyrimidin]-6'-one, 2'-chloro-7',8'-dihydro-Target API: Trilaciclib
C-21CAS 2231673-65-5
1-(3-Fluoropropyl)azetidin-3-amine bis(4-methylbenzenesulfonate)Target API: Camizestrant
C-22CAS 2222846-04-8
Carbamic acid, N-[(1R)-1-methyl-2-[1-(tetrahydro-2H-pyran-2-yl)-1H-indazol-4-yl]ethyl]-, 1,1-dimethylethyl esterTarget API: Camizestrant
C-23CAS 1690223-94-9
((S)-2-(2-MorpholinoacetaMido)-4-phenylbutanoyl)-L-leucyl-L-phenylalanineTarget API: carfilzomib
C-24CAS 1140908-89-9
(alphaS)-alpha-[[2-(4-Morpholinyl)acetyl]amino]benzenebutanoyl-L-leucyl-L-phenylalanine methyl esterTarget API: carfilzomib
C-26CAS 2222653-74-7
4-(6-Fluoropyridin-3-yl)-6-(2-hydroxy-2-methylpropoxy)pyrazolo[1,5-a]pyridine-3-carbonitrileTarget API: Selpercatinib
C-27CAS 2222654-09-1
4-(6-Fluoropyridin-3-yl)-6-hydroxypyrazolo[1,5-a]pyridine-3-carbonitrileTarget API: Selpercatinib
C-28CAS 869494-16-6
6-(tert-Butyloxycarbonyl)-3,6-diazabicyclo[3.1.1]heptaneTarget API: Selpercatinib
C-30CAS 1207836-10-9
6-bromo-4-methoxypyrazolo[1,5-a]pyridine-3-carbonitrileTarget API: Selpercatinib
C-32CAS 761440-65-7
1-(1-(3-Methoxy-4-nitrophenyl)piperidin-4-yl)-4-MethylpiperazineTarget API: Brigatinib
C-33CAS 761440-75-9
2-Methoxy-4-[4-(4-methylpiperazin-1-yl)piperidin-1-yl]anilineTarget API: Brigatinib
C-34CAS 1197953-49-3
25-Dichloro-N-[2-(dimethylphosphinyl)phenyl]-4-pyrimidinamineTarget API: Brigatinib
C-36CAS 1269440-69-8
CarbaMic acid,N-[5-chloro-2-fluoro-3-(4,4,5,5-tetramethyl-1,3,2-dioxaborolan-2-yl)phenyl]-, 1,1-dimethylethyl esterTarget API: Encorafenib
C-42CAS 3033111-52-0
(R)-6-(2-(ethylamino)-4-methoxyphenyl)-5,6,7,8-tetrahydronaphthalen-2-olTarget API: Elacestrant
C-44CAS 3057421-86-7
{2-[6-(benzyloxy)-3,4-dihydro-2-naphthyl]-5-methoxyphenyl}(ethyl)amineTarget API: Elacestrant
H-19CAS 1034975-62-6
4-(4-carboxy-3-(2,2,2-trifluoro-N-(tetrahydropyran-4-yl)acetamido)phenyl)-1-methylpiperazin-1-ium 2,2,2-trifluoroacetateTarget API: Entrectinib
