THERAPEUTIC AREA PORTFOLIO · 52 PRODUCTS

Oncology

肿瘤

Our oncology portfolio follows the terminal APIs represented in the catalog, spanning kinase inhibitors, DNA-damage and cell-cycle programs, endocrine oncology, and building blocks for ADC and PROTAC development.

Target APIs & Active Pipeline Programs in Oncology
SelpercatinibCapmatinibBrigatinibElacestrantEntrectinibNiraparibTrilaciclibCamizestrantCapivasertibCarfilzomibEncorafenibPalbociclibAbemaciclibAdagrasibLorlatinibOsimertinibRibociclibSotorasibADC PayloadADC LinkerPROTAC Linker

Oncology Products (52)

Catalog products related to terminal APIs in this area.

C-01APICAS 1231929-97-7
Abemaciclib
Target API: Abemaciclib
C-02APICAS 2326521-71-3
Adagrasib
Target API: Adagrasib
C-03CAS 1197377-47-1
(3-Amino-1,2,4-triazin-6-yl)-2-fluorobenzonitrile
Target API: Capmatinib
C-04CAS 870238-67-8
8-Cyano-3-fluorophenylboronic acid pinacol ester
Target API: Capmatinib
C-05CAS 69249-22-5
Amino-6-bromo-1,2,4-triazine
Target API: Capmatinib
C-07APICAS 1454846-35-5
Lorlatinib
Target API: Lorlatinib
C-08CAS 1171197-20-8
(S)-tert-butyl 3-(4-aminophenyl)piperidine-1-carboxylate
Target API: Niraparib
C-09CAS 138229-59-1
Methyl 3-formyl-2-nitrobenzoate
Target API: Niraparib
C-10CAS 875798-79-1
tert-Butyl 3-(4-Aminophenyl)piperidine-1-carboxylate
Target API: Niraparib
C-11APICAS 1421373-65-0
Osimertinib
Target API: Osimertinib
C-13CAS 571188-59-5
tert-butyl 4-(6-aminopyridin-3-yl)piperazine-1-carboxylate
Target API: Palbociclib
C-14APICAS 1211441-98-3
Ribociclib
Target API: Ribociclib
C-15APICAS 2296729-00-3
Sotorasib
Target API: Sotorasib
C-16CAS 571189-49-6
1-Methyl-4-(6-aminopyridin-3-yl)Piperazine
Target API: Trilaciclib
C-17CAS 36082-50-5
5-Bromo-2,4-dichloropyrimidine
Target API: Trilaciclib
C-19CAS 886061-26-3
(S)-3-(4-CHLOROPHENYL)-BETA-ALANINOL
Target API: Capivasertib
C-20CAS 252720-31-3
N-BOC-AMINO-PIPERIDINYL-1,1-CARBOXYLIC ACID
Target API: Capivasertib
C-25CAS 773-64-8
2-Mesitylenesulfonyl chloride
Target API: Selpercatinib
C-28CAS 869494-16-6
6-(tert-Butyloxycarbonyl)-3,6-diazabicyclo[3.1.1]heptane
Target API: Selpercatinib
C-29CAS 65873-72-5
6-Methoxy-3-pyridinecarboxaldehyde
Target API: Selpercatinib
C-30CAS 1207836-10-9
6-bromo-4-methoxypyrazolo[1,5-a]pyridine-3-carbonitrile
Target API: Selpercatinib
C-31CAS 36016-38-3
tert-Butyl N-hydroxycarbamate; N-Boc-hydroxylamine
Target API: Selpercatinib
C-35CAS 1229025-32-4
(S)-Methyl 1-aminopropan-2-ylcarbamate hydrochloride
Target API: Encorafenib
C-43CAS 722536-73-4
7-(benzyloxy)-3-bromo-1,2-dihydronaphthalene
Target API: Elacestrant
G-01CAS 159857-80-4
MC-Val-Cit-PABCMC---PABC
Target API: ADC Linker
G-02CAS 64987-85-5
SMCCSMCC-4-(N-)-1-
Target API: ADC Linker
G-03CAS 197720-53-9
Exatecan mesylate
Target API: ADC Payload
G-04CAS 1599440-33-1
DXd (Exatecan derivative)DXd
Target API: ADC Payload
G-05CAS 474645-27-7
MMAE (Monomethyl auristatin E)MMAEE
Target API: ADC Payload
G-06CAS 745017-94-1
MMAF (Monomethyl auristatin F)MMAFF
Target API: ADC Payload
G-07CAS 1594094-64-0
PBD Dimer (SG3199)PBDSG3199
Target API: ADC Payload
G-08CAS 86639-52-3
SN-38SN-38
Target API: ADC Payload
G-09CAS 1835736-39-4
Thalidomide-NH-PEG4-COOH-NH-PEG4-COOH
Target API: PROTAC Linker
G-10CAS 2098836-45-2
VH032-PEG4-COOHVH032-PEG4-COOH
Target API: PROTAC Linker
H-20CAS 1108745-30-7
5-(3,5-difluorobenzyl)-1H-indazol-3-amine
Target API: Entrectinib
H-21CAS 1108745-25-0
5-(3,5-difluorobenzyl)-2-fluorobenzonitrile
Target API: Entrectinib